Organic & Biomolecular Chemistry Blog

Pd(0)-catalyzed benzylic arylation–oxidation of 4-methylquinazolines via sp3 C–H activation under air conditions
Dan Zhao, Min-Xue Zhu, Yue Wang, Qi Shen and Jian-Xin Li
Org. Biomol. Chem., 2013,11, 6246-6249
DOI: 10.1039/C3OB41488D, Communication 

Major mechanistic differences between the reactions of hydroxylamine with phosphate di- and tri-esters
Michelle Medeiros, Eduardo H. Wanderlind, José R. Mora, Raphaell Moreira, Anthony J. Kirby and Faruk Nome
Org. Biomol. Chem., 2013,11, 6272-6284
DOI: 10.1039/C3OB40988K, Paper
From themed collection In Celebration of Andrew D. Hamilton’s Career in Chemistry  

Novel synthesis of various orthogonally protected Cα-methyllysine analogues and biological evaluation of a Vapreotide analogue containing (S)-α-methyllysine
Souvik Banerjee, Walker J. Wiggins, Jessie L. Geoghegan, Catherine T. Anthony, Eugene A. Woltering and Douglas S. Masterson
Org. Biomol. Chem., 2013,11, 6307-6319
DOI: 10.1039/C3OB41282B, Paper

Synthesis of novel pyrazole-based heterocycles via a copper(II)-catalysed domino annulation
Márió Gyuris, László G. Puskás, Gábor K. Tóth and Iván Kanizsai
Org. Biomol. Chem., 2013,11, 6320-6327
DOI: 10.1039/C3OB41146J, Paper

Structure–activity studies of 4-phenyl-substituted 2′-benzoylpyridine thiosemicarbazones with potent and selective anti-tumour activity
Adeline Y. Lukmantara, Danuta S. Kalinowski, Naresh Kumar and Des R. Richardson
Org. Biomol. Chem., 2013,11, 6414-6425
DOI: 10.1039/C3OB41109E, Paper

Bifunctional building blocks in the Ugi-azide condensation reaction: a general strategy toward exploration of new molecular diversity
Steven Gunawan and Christopher Hulme
Org. Biomol. Chem., 2013, Advance Article
DOI: 10.1039/C3OB40900G, Paper 

Comparative in vitro studies of MR imaging probes for metabotropic glutamate subtype-5 receptor targeting
Sven Gottschalk, Jörn Engelmann, Gabriele A. Rolla, Mauro Botta, David Parker and Anurag Mishra
Org. Biomol. Chem., 2013, Advance Article
DOI: 10.1039/C3OB41297K, Paper 

Synthesis and biological evaluation of non-isomerizable analogues of Ala-tRNA^Ala
Denia Mellal, Matthieu Fonvielle, Marco Santarem, Maryline Chemama, Yoann Schneider, Laura Iannazzo, Emmanuelle Braud, Michel Arthur and Mélanie Etheve-Quelquejeu
Org. Biomol. Chem., 2013, Advance Article
DOI: 10.1039/C3OB41206G, Paper 

First synthesis of antitumoral dasyscyphin B
Ali Akhaouzan, Antonio Fernández, Ahmed I. Mansour, Esteban Alvarez, Ali Haidöur, Ramón Alvarez-Manzaneda, Rachid Chahboun and Enrique Alvarez-Manzaneda
Org. Biomol. Chem., 2013, Advance Article
DOI: 10.1039/C3OB41290C, Paper                                          

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